BX795 is a potent and specific PDK1 inhibitor with IC50 of 6 nM, 140- and 1600-fold more selective for PDK1 than PKA and PKC, respectively. Meanwhile, in comparison to GSK3¦Â more than 100-fold selectivity observed for PDK1.

prudect name : BX795 is a potent and specific PDK1 inhibitor with IC50 of 6 nM, 140- and 1600-fold more selective for PDK1 than PKA and PKC, respectively. Meanwhile, in comparison to GSK3¦Â more than 100-fold selectivity observed for PDK1.
BX795 BX-795

Synonyms: CAS NO: 702675-74-9Molecular Formula: C₂₀H₂₃BrN₈OMolecular Weight: 471.36Purity: 98% minSolubility: In DMSOStorage: -20°C

162635-04-3 References PubMed ID：:http://www.ncbi.nlm.nih.gov/pubmed/1850335